Hotline:400-820-3792Inhibitors?ScreeningLibraries?Proteinswww.MedChemEMAT2Ainhibitor1Cat.No.:HY-112131CASNo.:2201057-10-3分?式:C??H??N?OS分?量:526.61作?靶點:MethionineAdenosyltransferase(MAT)作?通路:Epigenetics;MetabolicEnzyme/Protease儲存?式:Powder-20°C3years4°C2yearsInsolvent-80°C6months-20°C1month溶解性數(shù)據(jù)體外實驗DMSO:5mg/mL(9.49mM;Needultrasonicandwarming)MassSolvent1mg5mg10mgConcentration制備儲備液1mM1.8989mL9.4947mL18.9894mL5mM0.3798mL1.8989mL3.7979mL10mM---------請根據(jù)產(chǎn)品在不同溶劑中的溶解度選擇合適的溶劑配制儲備液；?旦配成溶液，請分裝保存，避免反復(fù)凍融造成的產(chǎn)品失效。儲備液的保存?式和期限：-80°C,6months;-20°C,1month。-80°C儲存時，請在6個?內(nèi)使?，-20°C儲存時，請在1個?內(nèi)使?。BIOLOGICALACTIVITY?物活性MAT2Ainhibitor1甲硫氨酸腺苷轉(zhuǎn)移酶2A(MATA2)抑制劑，其IC50值?于100nM。IC50&TargetMATA2[1]體外研究MAT2Ainhibitor1(Compound196)isasafeandeffectivecompoundthatpreventsandmanagescancers1/2MasterofBioactiveMolecules—您?邊的抑制劑?師www.MedChemEwhilereducingoravoidingthetoxicitiesand/orsideeffectsassociatedwiththeconventionaltherapies.Thecancersincludethosethatarerefractorytostandardtreatments,suchassurgery,radiationtherapy,chemotherapyandhormonaltherapy[1].REFERENCES[1].ZenonD,etal.Inhibitorsofcellularmetabolicprocesses.08March2018.WO2018045071A1.McePdfHeightCaution:Producthasnotbeenfullyvalidatedformedicalapplications.Forresearchuseonly.Tel:400-820-3792ax:021-5